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6TDC

PPAR gamma ligand binding domain in complex with MRL-871

Summary for 6TDC
Entry DOI10.2210/pdb6tdc/pdb
DescriptorPeroxisome proliferator-activated receptor gamma, 4-{1-[2-chloro-6-(trifluoromethyl)benzoyl]-1H-indazol-3-yl}benzoic acid, GLYCEROL, ... (4 entities in total)
Functional Keywordsnuclear receptor, nr1c3, transcription factor, gene regulation
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight33836.45
Authors
de Vries, R.M.J.M.,Leijten-van de Gevel, I.A.,van Herk, K.H.N.,Brunsveld, L. (deposition date: 2019-11-08, release date: 2020-11-18, Last modification date: 2024-01-24)
Primary citationLeijten-van de Gevel, I.A.,van Herk, K.H.N.,de Vries, R.M.J.M.,Brunsveld, L.
Binding of PPAR(gamma) to MRL871
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.328 Å)
Structure validation

237423

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