6QCK
17beta-hydroxysteroid dehydrogenase 14 variant T205 in complex with FB262
Summary for 6QCK
Entry DOI | 10.2210/pdb6qck/pdb |
Descriptor | 17-beta-hydroxysteroid dehydrogenase 14, DIMETHYL SULFOXIDE, 2-[2-(1,3-benzodioxol-2-yl)ethyl]benzoic acid, ... (7 entities in total) |
Functional Keywords | fragments, soaking, 17b-hsd14, oxidoreductase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 29897.72 |
Authors | Bertoletti, N.,Marchais-Oberwinkler, S.,Heine, A.,Klebe, G. (deposition date: 2018-12-28, release date: 2020-01-29, Last modification date: 2024-01-24) |
Primary citation | Badran, M.J.,Bertoletti, N.,Keils, A.,Heine, A.,Klebe, G.,Marchais-Oberwinkler, S. Mutational and structural studies uncover crucial amino acids determining activity and stability of 17 beta-HSD14. J.Steroid Biochem.Mol.Biol., 189:135-144, 2019 Cited by PubMed: 30836176DOI: 10.1016/j.jsbmb.2019.02.009 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.68 Å) |
Structure validation
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