6MNH
ULK1 Unc-51 like autophagy activating kinase in complex with inhibitor BTC
Summary for 6MNH
Entry DOI | 10.2210/pdb6mnh/pdb |
Descriptor | Serine/threonine-protein kinase ULK1, N-[(2R)-3-methylbutan-2-yl]-1H-benzotriazole-6-carboxamide, DIMETHYL SULFOXIDE, ... (5 entities in total) |
Functional Keywords | kinase, inhibitor, complex, transferase, transferase-inhibitor complex, transferase/inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 32937.99 |
Authors | Hendle, J.,Sauder, J.M.,Hickey, M.J.,Rauch, C.T.,Maletic, M.,Schwinn, K.D. (deposition date: 2018-10-01, release date: 2019-03-27, Last modification date: 2019-11-13) |
Primary citation | Nicolaou, C.A.,Humblet, C.,Hu, H.,Martin, E.M.,Dorsey, F.C.,Castle, T.M.,Burton, K.I.,Hu, H.,Hendle, J.,Hickey, M.J.,Duerksen, J.,Wang, J.,Erickson, J.A. Idea2Data: Toward a New Paradigm for Drug Discovery. Acs Med.Chem.Lett., 10:278-286, 2019 Cited by PubMed: 30891127DOI: 10.1021/acsmedchemlett.8b00488 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.73 Å) |
Structure validation
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