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6GR8

Human AURKC INCENP complex bound to BRD-7880

Summary for 6GR8
Entry DOI10.2210/pdb6gr8/pdb
DescriptorAurora kinase C, Inner centromere protein, 1-[(2~{R},3~{S})-2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-3-methyl-6-oxidanylidene-5-[(2~{S})-1-oxidanylpropan-2-yl]-3,4-dihydro-2~{H}-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)urea, ... (4 entities in total)
Functional Keywordskinase, structural genomics consortium, sgc, transferase
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains2
Total formula weight41060.17
Authors
Abdul Azeez, K.R.,Sorrell, F.J.,von Delft, F.,Bountra, C.,Knapp, S.,Edwards, A.M.,Arrowsmith, C.,Elkins, J.M. (deposition date: 2018-06-10, release date: 2019-05-15, Last modification date: 2024-01-17)
Primary citationAbdul Azeez, K.R.,Elkins, J.M.
AURKC INCENP complex bound to BRD-7880
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.75 Å)
Structure validation

217705

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