Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

6F8T

Crystal structure of the PDE4D catalytic domain in complex with GEBR-4a

Summary for 6F8T
Entry DOI10.2210/pdb6f8t/pdb
DescriptorcAMP-specific 3',5'-cyclic phosphodiesterase 4D, ZINC ION, MAGNESIUM ION, ... (5 entities in total)
Functional Keywordspde4, catalytic domain, inhibitor, gebr, hydrolase
Biological sourceHomo sapiens (Human)
Cellular locationApical cell membrane : Q08499
Total number of polymer chains2
Total formula weight80315.26
Authors
Prosdocimi, T.,Donini, S.,Parisini, E. (deposition date: 2017-12-13, release date: 2018-05-16, Last modification date: 2024-01-17)
Primary citationProsdocimi, T.,Mollica, L.,Donini, S.,Semrau, M.S.,Lucarelli, A.P.,Aiolfi, E.,Cavalli, A.,Storici, P.,Alfei, S.,Brullo, C.,Bruno, O.,Parisini, E.
Molecular Bases of PDE4D Inhibition by Memory-Enhancing GEBR Library Compounds.
Biochemistry, 57:2876-2888, 2018
Cited by
PubMed: 29652483
DOI: 10.1021/acs.biochem.8b00288
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.8 Å)
Structure validation

217157

PDB entries from 2024-03-13

PDB statisticsPDBj update infoContact PDBjnumon