6EY7
Human cytomegalovirus terminase nuclease domain, Mn soaked, inhibitor bound
Summary for 6EY7
Entry DOI | 10.2210/pdb6ey7/pdb |
Descriptor | UL89 HCMV terminase, MANGANESE (II) ION, 4-[(4-fluorophenyl)methyl-methyl-amino]-2,4-bis(oxidanylidene)butanoic acid, ... (5 entities in total) |
Functional Keywords | cytomegalovirus, ul89, terminase, inhibitors, drug design, raltegravir, viral protein |
Biological source | Human herpesvirus 5 strain AD169 |
Total number of polymer chains | 4 |
Total formula weight | 128869.29 |
Authors | Bongarzone, S.,Nadal, M.,Kaczmarska, Z.,Machon, C.,Alvarez, M.,Albericio, F.,Coll, M. (deposition date: 2017-11-10, release date: 2018-10-03, Last modification date: 2024-01-17) |
Primary citation | Bongarzone, S.,Nadal, M.,Kaczmarska, Z.,Machon, C.,Alvarez, M.,Albericio, F.,Coll, M. Structure-Driven Discovery of alpha , gamma-Diketoacid Inhibitors Against UL89 Herpesvirus Terminase. Acs Omega, 3:8497-8505, 2018 Cited by PubMed: 31458978DOI: 10.1021/acsomega.8b01472 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.9 Å) |
Structure validation
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