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6CBZ

Estrogen Receptor Alpha Ligand Binding Domain Y537S Mutant in Complex with Estradiol and GRIP Peptide

Summary for 6CBZ
Entry DOI10.2210/pdb6cbz/pdb
DescriptorEstrogen receptor, grip peptide, ESTRADIOL, ... (6 entities in total)
Functional Keywordsbreast cancer, steroid receptor, estrogen, hormone, transcription
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains4
Total formula weight59572.42
Authors
Fanning, S.W.,Greene, G.L. (deposition date: 2018-02-05, release date: 2018-02-28, Last modification date: 2020-02-26)
Primary citationMaximov, P.Y.,Abderrahman, B.,Fanning, S.W.,Sengupta, S.,Fan, P.,Curpan, R.F.,Rincon, D.M.Q.,Greenland, J.A.,Rajan, S.S.,Greene, G.L.,Jordan, V.C.
Endoxifen, 4-Hydroxytamoxifen and an Estrogenic Derivative Modulate Estrogen Receptor Complex Mediated Apoptosis in Breast Cancer.
Mol. Pharmacol., 94:812-822, 2018
Cited by
PubMed: 29739819
DOI: 10.1124/mol.117.111385
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.65 Å)
Structure validation

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