6CBZ
Estrogen Receptor Alpha Ligand Binding Domain Y537S Mutant in Complex with Estradiol and GRIP Peptide
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 7 |
Details | binding site for residue EST A 601 |
Chain | Residue |
A | MET343 |
A | LEU346 |
A | GLU353 |
A | ARG394 |
A | HIS524 |
A | LEU525 |
A | HOH807 |
site_id | AC2 |
Number of Residues | 7 |
Details | binding site for residue GOL B 601 |
Chain | Residue |
B | LEU408 |
B | LEU409 |
B | LEU410 |
B | GLN414 |
B | HOH701 |
B | PHE337 |
B | ASN407 |
site_id | AC3 |
Number of Residues | 6 |
Details | binding site for residue EST B 602 |
Chain | Residue |
B | LEU346 |
B | GLU353 |
B | ARG394 |
B | HIS524 |
B | LEU525 |
B | HOH759 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 1 |
Details | MOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106 |
Chain | Residue | Details |
B | SER537 |
site_id | SWS_FT_FI2 |
Number of Residues | 1 |
Details | LIPID: S-palmitoyl cysteine => ECO:0000250 |
Chain | Residue | Details |
B | CYS447 |