6Z52
Crystal structure of CLK3 in complex with macrocycle ODS2003136
Summary for 6Z52
Entry DOI | 10.2210/pdb6z52/pdb |
Descriptor | Dual specificity protein kinase CLK3, 1,2-ETHANEDIOL, CHLORIDE ION, ... (6 entities in total) |
Functional Keywords | kinase, kinase inhibitor, clk3, macrocycle, nanocyclic, structural genomics, structural genomics consortium, sgc, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 88133.16 |
Authors | Chaikuad, A.,Benderitter, P.,Hoflack, J.,Denis, A.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2020-05-26, release date: 2020-06-03, Last modification date: 2024-01-24) |
Primary citation | Chaikuad, A.,Benderitter, P.,Hoflack, J.,Denis, A.,Knapp, S.,Structural Genomics Consortium (SGC) Crystal structure of CLK3 in complex with macrocycle ODS2003136 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.12 Å) |
Structure validation
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