6XVF
Crystal structure of bovine cytochrome bc1 in complex with tetrahydro-quinolone inhibitor JAG021
Summary for 6XVF
Entry DOI | 10.2210/pdb6xvf/pdb |
Descriptor | Cytochrome b-c1 complex subunit 1, mitochondrial, Cytochrome b-c1 complex subunit 9, TETRAETHYLENE GLYCOL, ... (22 entities in total) |
Functional Keywords | cytochrome bc1, malaria, electron transport, membrane protein |
Biological source | Bos taurus (cattle) More |
Total number of polymer chains | 10 |
Total formula weight | 238215.60 |
Authors | Amporndanai, K.,Hasnain, S.S.,Antonyuk, S.V. (deposition date: 2020-01-21, release date: 2020-07-22, Last modification date: 2024-01-24) |
Primary citation | McPhillie, M.J.,Zhou, Y.,Hickman, M.R.,Gordon, J.A.,Weber, C.R.,Li, Q.,Lee, P.J.,Amporndanai, K.,Johnson, R.M.,Darby, H.,Woods, S.,Li, Z.H.,Priestley, R.S.,Ristroph, K.D.,Biering, S.B.,El Bissati, K.,Hwang, S.,Hakim, F.E.,Dovgin, S.M.,Lykins, J.D.,Roberts, L.,Hargrave, K.,Cong, H.,Sinai, A.P.,Muench, S.P.,Dubey, J.P.,Prud'homme, R.K.,Lorenzi, H.A.,Biagini, G.A.,Moreno, S.N.,Roberts, C.W.,Antonyuk, S.V.,Fishwick, C.W.G.,McLeod, R. Potent Tetrahydroquinolone Eliminates Apicomplexan Parasites. Front Cell Infect Microbiol, 10:203-203, 2020 Cited by PubMed: 32626661DOI: 10.3389/fcimb.2020.00203 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.5 Å) |
Structure validation
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