6W1Y
Cryo-EM structure of 5HT3A receptor in presence of Palonosetron
Summary for 6W1Y
Entry DOI | 10.2210/pdb6w1y/pdb |
EMDB information | 21511 21512 21518 |
Descriptor | 5-hydroxytryptamine receptor 3A, 2-acetamido-2-deoxy-beta-D-glucopyranose-(4-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (5 entities in total) |
Functional Keywords | transport protein |
Biological source | Mus musculus (Mouse) |
Total number of polymer chains | 5 |
Total formula weight | 268869.36 |
Authors | |
Primary citation | Basak, S.,Kumar, A.,Ramsey, S.,Gibbs, E.,Kapoor, A.,Filizola, M.,Chakrapani, S. High-resolution structures of multiple 5-HT 3A R-setron complexes reveal a novel mechanism of competitive inhibition. Elife, 9:-, 2020 Cited by PubMed: 33063666DOI: 10.7554/eLife.57870 PDB entries with the same primary citation |
Experimental method | ELECTRON MICROSCOPY (3.35 Å) |
Structure validation
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