6NP0
Cryo-EM structure of 5HT3A receptor in presence of granisetron
Summary for 6NP0
Entry DOI | 10.2210/pdb6np0/pdb |
EMDB information | 0469 |
Descriptor | 5-hydroxytryptamine receptor 3A, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (6 entities in total) |
Functional Keywords | membrane protein |
Biological source | Mus musculus (Mouse) |
Total number of polymer chains | 5 |
Total formula weight | 290284.84 |
Authors | Basak, S.,Chakrapani, S. (deposition date: 2019-01-17, release date: 2019-07-24, Last modification date: 2020-07-29) |
Primary citation | Basak, S.,Gicheru, Y.,Kapoor, A.,Mayer, M.L.,Filizola, M.,Chakrapani, S. Molecular mechanism of setron-mediated inhibition of full-length 5-HT3Areceptor. Nat Commun, 10:3225-3225, 2019 Cited by PubMed: 31324772DOI: 10.1038/s41467-019-11142-8 PDB entries with the same primary citation |
Experimental method | ELECTRON MICROSCOPY (2.92 Å) |
Structure validation
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