6EHA
Heme oxygenase 1 in complex with inhibitor
Summary for 6EHA
Entry DOI | 10.2210/pdb6eha/pdb |
Descriptor | Heme oxygenase 1, PROTOPORPHYRIN IX CONTAINING FE, 1-(3-imidazol-1-ylpropyl)-5-(2-methylpropyl)-4-phenyl-imidazole, ... (4 entities in total) |
Functional Keywords | heme oxygenase, oxidoreductase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 67570.93 |
Authors | Grudnik, P.,Mieczkowski, M. (deposition date: 2017-09-12, release date: 2018-10-10, Last modification date: 2024-05-08) |
Primary citation | Mucha, O.,Podkalicka, P.,Mikulski, M.,Barwacz, S.,Andrysiak, K.,Biela, A.,Mieczkowski, M.,Kachamakova-Trojanowska, N.,Ryszawy, D.,Bialas, A.,Szelazek, B.,Grudnik, P.,Majewska, E.,Michalik, K.,Jakubiec, K.,Bien, M.,Witkowska, N.,Gluza, K.,Ekonomiuk, D.,Sitarz, K.,Galezowski, M.,Brzozka, K.,Dubin, G.,Jozkowicz, A.,Dulak, J.,Loboda, A. Development and characterization of a new inhibitor of heme oxygenase activity for cancer treatment. Arch.Biochem.Biophys., 671:130-142, 2019 Cited by PubMed: 31276659DOI: 10.1016/j.abb.2019.07.002 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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