6BS0
JAK2 JH2 in complex with 63552444
Summary for 6BS0
Entry DOI | 10.2210/pdb6bs0/pdb |
Descriptor | Tyrosine-protein kinase JAK2, 4-(5-aminopyrazin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine, GLYCEROL, ... (4 entities in total) |
Functional Keywords | pseudokinase domain, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 33623.48 |
Authors | Puleo, D.E.,Schlessinger, J. (deposition date: 2017-12-01, release date: 2018-08-22, Last modification date: 2023-10-04) |
Primary citation | Puleo, D.E.,Schlessinger, J. JAK2 JH2 Binders To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.541 Å) |
Structure validation
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