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6BS0

JAK2 JH2 in complex with 63552444

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue E4V A 901
ChainResidue
ALEU551
AHOH1021
AHOH1064
AHOH1180
AILE559
ALEU579
AGLU627
APHE628
AVAL629
ALYS630
AGLY632
ALEU680

site_idAC2
Number of Residues5
Detailsbinding site for residue GOL A 902
ChainResidue
AASN673
ATRP718
AHOH1001
AHOH1015
AHOH1069

site_idAC3
Number of Residues8
Detailsbinding site for residue GOL A 903
ChainResidue
AGLN771
AASN785
AMET788
AASP789
AHOH1079
AHOH1083
AHOH1098
AHOH1162

site_idAC4
Number of Residues4
Detailsbinding site for residue GOL A 904
ChainResidue
APHE694
AHOH1012
AHOH1106
AHOH1187

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Breakpoint for translocation to form PCM1-JAK2 fusion protein
ChainResidueDetails
AASP710

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphotyrosine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ATYR570

222415

PDB entries from 2024-07-10

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