5XHK
Crystal structure of the BRD2-BD2 in complex with phenanthridinone
Summary for 5XHK
| Entry DOI | 10.2210/pdb5xhk/pdb |
| Related | 5XHE |
| Descriptor | Bromodomain-containing protein 2, GLYCEROL, METHOXYETHANE, ... (5 entities in total) |
| Functional Keywords | bromodomain, bet family, brd2, phenanthridinone, transcription |
| Biological source | Homo sapiens (Human) |
| Total number of polymer chains | 1 |
| Total formula weight | 13845.82 |
| Authors | Padmanabhan, B.,Mathur, S.,Tripathi, S.,Deshmukh, P. (deposition date: 2017-04-21, release date: 2017-09-06, Last modification date: 2023-11-22) |
| Primary citation | Mathur, S.,Deshmukh, P.,Tripathi, S.,Marimuthu, P.,Padmanabhan, B. Insights into the crystal structure of BRD2-BD2 - phenanthridinone complex and theoretical studies on phenanthridinone analogs. J. Biomol. Struct. Dyn., 36:2342-2360, 2018 Cited by PubMed: 28696179DOI: 10.1080/07391102.2017.1353441 PDB entries with the same primary citation |
| Experimental method | X-RAY DIFFRACTION (1.28 Å) |
Structure validation
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