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5XHK

Crystal structure of the BRD2-BD2 in complex with phenanthridinone

Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue GOL A 501
ChainResidue
ATYR368
ALYS402
AASP407
AMET438
ALYS441
AHOH607
AHOH617
AHOH662

site_idAC2
Number of Residues6
Detailsbinding site for residue GOL A 502
ChainResidue
ATYR373
AHOH601
AHOH602
AHOH668
AHOH728
ALEU361

site_idAC3
Number of Residues4
Detailsbinding site for residue 2ME A 503
ChainResidue
ATRP370
AVAL435
AMET438
ALDR504

site_idAC4
Number of Residues8
Detailsbinding site for residue LDR A 504
ChainResidue
APRO371
AVAL376
ALEU381
ALEU383
ACYS425
AASN429
A2ME503
AHOH604

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues109
DetailsDomain: {"description":"Bromo 2","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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