5US1
Crystal structure of aminoglycoside acetyltransferase AAC(2')-Ia in complex with N2'-acetylgentamicin C1A and coenzyme A
Summary for 5US1
Entry DOI | 10.2210/pdb5us1/pdb |
Related | 6C0C |
Descriptor | Aminoglycoside 2'-N-acetyltransferase, (1R,2S,3S,4R,6S)-4,6-diamino-3-{[3-deoxy-4-C-methyl-3-(methylamino)-beta-L-arabinopyranosyl]oxy}-2-hydroxycyclohexyl 2-(acetylamino)-6-amino-2,3,4,6-tetradeoxy-alpha-D-erythro-hexopyranoside, D(-)-TARTARIC ACID, ... (7 entities in total) |
Functional Keywords | gnat, gcn5-n-acetyltransferase, acetyltransferase, aminoglycoside, gentamicin, coenzyme a, acetylcoenzyme a antibiotic resistance, structural genomics, center for structural genomics of infectious diseases, csgid, national institute of allergy and infectious diseases, niaid, transferase |
Biological source | Providencia stuartii |
Total number of polymer chains | 12 |
Total formula weight | 263334.07 |
Authors | Stogios, P.J.,Evdokimova, E.,Xu, Z.,Wawrzak, Z.,Savchenko, A.,Anderson, W.F.,Center for Structural Genomics of Infectious Diseases (CSGID) (deposition date: 2017-02-13, release date: 2017-03-15, Last modification date: 2023-10-04) |
Primary citation | Cox, G.,Ejim, L.,Stogios, P.J.,Koteva, K.,Bordeleau, E.,Evdokimova, E.,Sieron, A.O.,Savchenko, A.,Serio, A.W.,Krause, K.M.,Wright, G.D. Plazomicin Retains Antibiotic Activity against Most Aminoglycoside Modifying Enzymes. ACS Infect Dis, 4:980-987, 2018 Cited by PubMed: 29634241DOI: 10.1021/acsinfecdis.8b00001 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.48 Å) |
Structure validation
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