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5OML

Crystal structure of Trypanosoma Brucei PEX14 N-terminal domain in complex with small molecules to investigate the water envelope

Summary for 5OML
Entry DOI10.2210/pdb5oml/pdb
DescriptorPeroxin 14, (3~{R})-3-[[1-(2-hydroxyethyl)-5-[(4-methoxynaphthalen-1-yl)methyl]-6,7-dihydro-4~{H}-pyrazolo[4,3-c]pyridin-3-yl]carbonylamino]-3-phenyl-propanoic acid, SULFATE ION, ... (5 entities in total)
Functional Keywordsperoxisomal translocation, ppi inhibition, protein-inhibitor complex, signaling protein
Biological sourceTrypanosoma brucei brucei
Total number of polymer chains4
Total formula weight33927.02
Authors
Ratkova, E.L.,Dawidowski, M.,Napolitano, V.,Dubin, G.,Fino, R.,Popowicz, G.,Sattler, M.,Tetko, I.V. (deposition date: 2017-08-01, release date: 2019-03-06, Last modification date: 2024-01-17)
Primary citationRatkova, E.L.,Dawidowski, M.,Napolitano, V.,Dubin, G.,Fino, R.,Popowicz, G.,Sattler, M.,Tetko, I.V.
Crystal structure of Trypanosoma Brucei PEX14 N-terminal domain in complex with small molecules to investigate the water envelope
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.5 Å)
Structure validation

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