5KO1
Pseudokinase Domain of MLKL bound to Compound 4.
Summary for 5KO1
Entry DOI | 10.2210/pdb5ko1/pdb |
Related | 5KNJ |
Descriptor | Mixed lineage kinase domain-like protein, [(1~{R})-2-[(4-fluorophenyl)amino]-2-oxidanylidene-1-phenyl-ethyl] 3-azanylpyrazine-2-carboxylate (3 entities in total) |
Functional Keywords | pseudokinase domain mlkl type1 inhibitor, membrane proteins-inhibitor complex, membrane proteins/inhibitor |
Biological source | Homo sapiens (Human) |
Cellular location | Cytoplasm : Q8NB16 |
Total number of polymer chains | 1 |
Total formula weight | 32599.51 |
Authors | Marcotte, D.J. (deposition date: 2016-06-29, release date: 2016-11-16, Last modification date: 2023-09-27) |
Primary citation | Ma, B.,Marcotte, D.,Paramasivam, M.,Michelsen, K.,Wang, T.,Bertolotti-Ciarlet, A.,Jones, J.H.,Moree, B.,Butko, M.,Salafsky, J.,Sun, X.,McKee, T.,Silvian, L.F. ATP-Competitive MLKL Binders Have No Functional Impact on Necroptosis. Plos One, 11:e0165983-e0165983, 2016 Cited by PubMed: 27832137DOI: 10.1371/journal.pone.0165983 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.16 Å) |
Structure validation
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