5KH6

SETDB1 in complex with a fragment candidate

Summary for 5KH6

• Entry DOI: 10.2210/pdb5kh6/pdb
• Descriptor: Histone-lysine N-methyltransferase SETDB1, 1,2-ETHANEDIOL, DIMETHYL SULFOXIDE, ... (10 entities in total)
• Functional Keywords: fragment screening, structural genomics consortium, sgc, diamond i04-1 xchem, pandda, transferase
• Biological source: Homo sapiens (Human)
• Cellular location: Nucleus: Q15047
• Total number of polymer chains: 1
• Total formula weight: 26274.66

Authors

Walker, J.R.,Harding, R.J.,Mader, P.,Dobrovetsky, E.,Dong, A.,Collins, P.,Pearce, N.,Brandao-Neto, J.,Douangamath, A.,von Delft, F.,Brown, P.J.,Schapira, M.,Arrowsmith, C.H.,Edwards, A.M.,Santhakumar, V.,Structural Genomics Consortium (SGC) (deposition date: 2016-06-14, release date: 2016-09-21, Last modification date: 2024-04-03)

• Primary citation: Walker, J.R.,Harding, R.J.,Mader, P.,Dobrovetsky, E.,Dong, A.,Collins, P.,Pearce, N.,Brandao-Neto, J.,Douangamath, A.,von Delft, F.,Brown, P.J.,Schapira, M.,Arrowsmith, C.H.,Edwards, A.M.,Santhakumar, V.,Structural Genomics Consortium (SGC); SETDB1 in complex with a fragment candidate; To be published,

Experimental method

X-RAY DIFFRACTION (2.05 Å)