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5KH6

SETDB1 in complex with a fragment candidate

Functional Information from PDB Data
site_idAC1
Number of Residues3
Detailsbinding site for residue EDO A 501
ChainResidue
AGLN273
AVAL274
ATRP275

site_idAC2
Number of Residues5
Detailsbinding site for residue DMS A 502
ChainResidue
AGLY300
ATYR301
AGLU386
AARG394
A6SU513

site_idAC3
Number of Residues6
Detailsbinding site for residue EDO A 503
ChainResidue
ALYS208
ALYS211
ALEU242
AHIS246
AHOH693
ALYS207

site_idAC4
Number of Residues7
Detailsbinding site for residue SO4 A 504
ChainResidue
AHIS214
ALYS215
AHOH606
AHOH618
AHOH619
AHOH648
AHOH658

site_idAC5
Number of Residues4
Detailsbinding site for residue SO4 A 505
ChainResidue
AASP270
AGLY271
AASN272
AGLN273

site_idAC6
Number of Residues4
Detailsbinding site for residue SO4 A 506
ChainResidue
ATHR306
AGLN307
ASER308
AARG384

site_idAC7
Number of Residues3
Detailsbinding site for residue SO4 A 507
ChainResidue
AARG203
AHOH637
AHOH715

site_idAC8
Number of Residues3
Detailsbinding site for residue SO4 A 508
ChainResidue
APRO316
ALYS318
AHOH634

site_idAC9
Number of Residues3
Detailsbinding site for residue CL A 509
ChainResidue
AARG209
ALYS364
AASP381

site_idAD1
Number of Residues3
Detailsbinding site for residue CL A 510
ChainResidue
ALYS318
ASER350
AEDO514

site_idAD2
Number of Residues2
Detailsbinding site for residue CL A 511
ChainResidue
ASER243
AHIS246

site_idAD3
Number of Residues1
Detailsbinding site for residue CL A 512
ChainResidue
AGLY225

site_idAD4
Number of Residues9
Detailsbinding site for residue 6SU A 513
ChainResidue
APHE296
AGLY300
AALA302
ASER328
ACYS329
APHE332
ATYR389
ADMS502
AHOH660

site_idAD5
Number of Residues5
Detailsbinding site for residue EDO A 514
ChainResidue
AASN245
AARG315
APRO316
ALEU317
ACL510

site_idAD6
Number of Residues5
Detailsbinding site for residue PEG A 515
ChainResidue
ALYS269
ATYR301
AALA302
ATRP387
AHOH620

site_idAD7
Number of Residues8
Detailsbinding site for residue PEG A 516
ChainResidue
AGLU283
AASN286
ALYS288
ATYR304
AARG343
AGLY372
ASER373
AHOH719

site_idAD8
Number of Residues4
Detailsbinding site for residue PEG A 517
ChainResidue
ALYS290
AARG292
AASP371
AHOH724

site_idAD9
Number of Residues3
Detailsbinding site for residue ACT A 518
ChainResidue
AGLU190
AASN191
ATHR223

site_idAE1
Number of Residues6
Detailsbinding site for residue EDO A 519
ChainResidue
ASER303
ATYR304
AASP371
ATRP387
AHOH640
AHOH650

site_idAE2
Number of Residues5
Detailsbinding site for residue GOL A 520
ChainResidue
ALYS208
ATHR210
ATHR212
AHIS214
AHOH743

224004

PDB entries from 2024-08-21

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