5JSJ
Crystal structure of Spindlin1 bound to compound EML631
Summary for 5JSJ
Entry DOI | 10.2210/pdb5jsj/pdb |
Related | 5JSG |
Descriptor | Spindlin-1, [4-(2-pyrrolidin-1-ylethyl)piperidin-1-yl]-[4-[4-(2-pyrrolidin-1-ylethyl)piperidin-1-yl]carbonyl-3-[[4-(pyrrolidin-1-ylmethoxy)phenyl]amino]phenyl]methanone, MAGNESIUM ION, ... (5 entities in total) |
Functional Keywords | tudor domain, cell cycle |
Biological source | Homo sapiens (Human) |
Cellular location | Nucleus : Q9Y657 |
Total number of polymer chains | 2 |
Total formula weight | 52484.61 |
Authors | |
Primary citation | Bae, N.,Viviano, M.,Su, X.,Lv, J.,Cheng, D.,Sagum, C.,Castellano, S.,Bai, X.,Johnson, C.,Khalil, M.I.,Shen, J.,Chen, K.,Li, H.,Sbardella, G.,Bedford, M.T. Developing Spindlin1 small-molecule inhibitors by using protein microarrays Nat. Chem. Biol., 13:750-756, 2017 Cited by PubMed: 28504676DOI: 10.1038/nchembio.2377 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.348 Å) |
Structure validation
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