5GIE
Crystal structure of VDR in complex with DLAM-4P (P21 form)
Summary for 5GIE
Entry DOI | 10.2210/pdb5gie/pdb |
Related | 5GIC 5GID |
Descriptor | Vitamin D3 receptor, SRC1, (3R,5S)-5-[(2R)-2-[(1R,3aS,4E,7aR)-7a-methyl-4-[(2Z)-2-[(3S,5R)-2-methylidene-3,5-bis(oxidanyl)cyclohexylidene]ethylidene]-2,3,3a,5,6,7-hexahydro-1H-inden-1-yl]propyl]-3-methyl-3-oxidanyl-1-(4-phenylbutyl)pyrrolidin-2-one, ... (4 entities in total) |
Functional Keywords | nuclear receptor, transcription |
Biological source | Rattus norvegicus (Rat) More |
Total number of polymer chains | 4 |
Total formula weight | 61747.54 |
Authors | Asano, L.,Shimizu, T. (deposition date: 2016-06-23, release date: 2016-12-07, Last modification date: 2024-03-20) |
Primary citation | Asano, L.,Waku, T.,Abe, R.,Kuwabara, N.,Ito, I.,Yanagisawa, J.,Nagasawa, K.,Shimizu, T. Regulation of the vitamin D receptor by vitamin D lactam derivatives. Febs Lett., 590:3270-3279, 2016 Cited by PubMed: 27500498DOI: 10.1002/1873-3468.12348 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.387 Å) |
Structure validation
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