5DCZ

Tankyrase 2 complexed with a selective inhibitor

Summary for 5DCZ

• Entry DOI: 10.2210/pdb5dcz/pdb
• Descriptor: Tankyrase-2, ZINC ION, PHOSPHATE ION, ... (5 entities in total)
• Functional Keywords: transferase-transferase inhibitor complex, transferase/transferase inhibitor
• Biological source: Homo sapiens (Human)
• Cellular location: Cytoplasm: Q9H2K2
• Total number of polymer chains: 1
• Total formula weight: 26620.22

Authors

Shewchuk, L.M.,Muelbaier, M. (deposition date: 2015-08-24, release date: 2016-09-07, Last modification date: 2023-09-27)

• Primary citation: Muelbaier, M.,Shewchuk, L.M.; Discovery of a new tool compound with superior selectivity to interrogate the biology of Tankyrase; J.Med.Chem, 2015

Experimental method

X-RAY DIFFRACTION (2.23 Å)