Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

5DCZ

Tankyrase 2 complexed with a selective inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 1201
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC2
Number of Residues6
Detailsbinding site for residue PO4 A 1202
ChainResidue
AHOH1355
AARG977
AHIS979
AARG980
ALYS1067
AHOH1354

site_idAC3
Number of Residues14
Detailsbinding site for residue 59B A 1203
ChainResidue
APHE1030
AHIS1031
AGLY1032
ASER1033
AARG1047
AHIS1048
AALA1049
ATYR1060
AALA1062
ASER1068
ATYR1071
AILE1075
AGLU1138
AHOH1316

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092

222415

PDB entries from 2024-07-10

PDB statisticsPDBj update infoContact PDBjnumon