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5DCZ

Tankyrase 2 complexed with a selective inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 1201
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC2
Number of Residues6
Detailsbinding site for residue PO4 A 1202
ChainResidue
AHOH1355
AARG977
AHIS979
AARG980
ALYS1067
AHOH1354

site_idAC3
Number of Residues14
Detailsbinding site for residue 59B A 1203
ChainResidue
APHE1030
AHIS1031
AGLY1032
ASER1033
AARG1047
AHIS1048
AALA1049
ATYR1060
AALA1062
ASER1068
ATYR1071
AILE1075
AGLU1138
AHOH1316

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"O95271","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

238895

PDB entries from 2025-07-16

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