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5B1S

Crystal structure of Trypanosoma cruzi spermidine synthase in complex with 2-(2-fluorophenyl)ethanamine

Summary for 5B1S
Entry DOI10.2210/pdb5b1s/pdb
DescriptorSpermidine synthase, putative, 5'-[(S)-(3-AMINOPROPYL)(METHYL)-LAMBDA~4~-SULFANYL]-5'-DEOXYADENOSINE, 2-(2-fluorophenyl)ethanamine, ... (4 entities in total)
Functional Keywordspolyamine synthesis, transferase
Biological sourceTrypanosoma cruzi strain CL Brener
Total number of polymer chains4
Total formula weight138397.35
Authors
Amano, Y.,Tateishi, Y. (deposition date: 2015-12-17, release date: 2016-12-21, Last modification date: 2023-11-08)
Primary citationYoshino, R.,Yasuo, N.,Hagiwara, Y.,Ishida, T.,Inaoka, D.K.,Amano, Y.,Tateishi, Y.,Ohno, K.,Namatame, I.,Niimi, T.,Orita, M.,Kita, K.,Akiyama, Y.,Sekijima, M.
In silico, in vitro, X-ray crystallography, and integrated strategies for discovering spermidine synthase inhibitors for Chagas disease
Sci Rep, 7:6666-6666, 2017
Cited by
PubMed: 28751689
DOI: 10.1038/s41598-017-06411-9
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.58 Å)
Structure validation

217705

건을2024-03-27부터공개중

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