4YJV
THE KINASE DOMAIN OF HUMAN SPLEEN TYROSINE (SYK) IN COMPLEX WITH GTC000250
Summary for 4YJV
Entry DOI | 10.2210/pdb4yjv/pdb |
Descriptor | Tyrosine-protein kinase SYK, 3-[6-({4-[ethyl(1H-indazol-4-yl)amino]-5-fluoropyrimidin-2-yl}amino)-2,4-dihydro-1H-indazol-1-yl]propan-1-ol (3 entities in total) |
Functional Keywords | syk, non-receptor tyrosine kinase, spleen tyrosine kinase, transferase, phosphorylation, transferase-transferase inhibitor complex |
Biological source | Homo sapiens (Human) |
Cellular location | Cell membrane : P43405 |
Total number of polymer chains | 1 |
Total formula weight | 33259.10 |
Authors | Somers, D.O.,Neu, M.,Stuckey, J. (deposition date: 2015-03-03, release date: 2015-10-14, Last modification date: 2024-05-01) |
Primary citation | Somers, D.O.,Neu, M.,Stuckey, J. THE KINASE DOMAIN OF HUMAN SPLEEN TYROSINE (SYK) IN COMPLEX WITH GTC000250 to be published, |
Experimental method | X-RAY DIFFRACTION (1.652 Å) |
Structure validation
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