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4TRY

Structure of BACE1 complex with a HEA-type inhibitor

Summary for 4TRY
Entry DOI10.2210/pdb4try/pdb
Related4TRW 4TRZ
Related PRD IDPRD_002106
DescriptorBeta-secretase 1, GLU-ILE-TIH-THC-NVA (3 entities in total)
Functional Keywordshydrase proteinase converting, designed inhibitor, hydrase-inhibitor complex, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains6
Total formula weight131933.04
Authors
Akaji, K.,Teruya, K.,Akiyama, T.,Sanjho, A.,Yamashita, E.,Nakagawa, A. (deposition date: 2014-06-18, release date: 2015-07-29, Last modification date: 2023-11-08)
Primary citationAkaji, K.,Teruya, K.,Akiyama, T.,Sanjho, A.,Yamashita, E.,Nakagawa, A.
Structure of BACE1 complex with an anti-HMC-type inhibitor
to be published,
Experimental method
X-RAY DIFFRACTION (2.75 Å)
Structure validation

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