4QMW
MST3 IN COMPLEX WITH PP-121, 1-CYCLOPENTYL-3-(1H-PYRROLO[2,3-B]PYRIDIN-5-YL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE
Summary for 4QMW
Entry DOI | 10.2210/pdb4qmw/pdb |
Related | 4QML 4QMM 4QMN 4QMO 4QMP 4QMQ 4QMS 4QMT 4QMV 4QMX 4QMY 4QMZ 4QO9 |
Descriptor | SERINE/THREONINE-PROTEIN KINASE 24, 1-cyclopentyl-3-(1H-pyrrolo[2,3-b]pyridin-5-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine, 1,2-ETHANEDIOL, ... (5 entities in total) |
Functional Keywords | protein kinase, mst3, stk24, sterile 20-like kinase, atp-binding, nucleotide-binding, phosphoprotein, serine/threonine-transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm: Q9Y6E0 |
Total number of polymer chains | 1 |
Total formula weight | 35464.41 |
Authors | Olesen, S.H.,Watts, C.,Zhu, J.-Y.,Schonbrunn, E. (deposition date: 2014-06-16, release date: 2015-07-01, Last modification date: 2023-09-20) |
Primary citation | Olesen, S.H.,Zhu, J.Y.,Martin, M.P.,Schonbrunn, E. Discovery of Diverse Small-Molecule Inhibitors of Mammalian Sterile20-like Kinase 3 (MST3). Chemmedchem, 11:1137-1144, 2016 Cited by PubMed: 27135311DOI: 10.1002/cmdc.201600115 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.6 Å) |
Structure validation
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