Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

4QMT

MST3 in complex with HESPERADIN

Summary for 4QMT
Entry DOI10.2210/pdb4qmt/pdb
Related4QML 4QMM 4QMN 4QMO 4QMP 4QMQ 4QMR 4QMS 4QMU 4QMV 4QMW 4QMX 4QMY 4QMZ
DescriptorSerine/threonine-protein kinase 24, N-[2-OXO-3-((E)-PHENYL{[4-(PIPERIDIN-1-YLMETHYL)PHENYL]IMINO}METHYL)-2,6-DIHYDRO-1H-INDOL-5-YL]ETHANESULFONAMIDE, 1,2-ETHANEDIOL, ... (4 entities in total)
Functional Keywordsprotein kinase, mst3, stk24, sterile 20-like kinase, atp-binding, nucleotide-binding, phosphoprotein, serine/threonine-transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm: Q9Y6E0
Total number of polymer chains1
Total formula weight35602.66
Authors
Olesen, S.H.,Watts, C.,Zhu, J.-Y.,Schonbrunn, E. (deposition date: 2014-06-16, release date: 2015-07-01, Last modification date: 2023-09-20)
Primary citationOlesen, S.H.,Zhu, J.Y.,Martin, M.P.,Schonbrunn, E.
Discovery of Diverse Small-Molecule Inhibitors of Mammalian Sterile20-like Kinase 3 (MST3).
Chemmedchem, 11:1137-1144, 2016
Cited by
PubMed: 27135311
DOI: 10.1002/cmdc.201600115
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.5 Å)
Structure validation

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon