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4Q4M

tRNA-Guanine Transglycosylase (TGT) in Complex with 6-Amino-4-phenyl-1,2-dihydro-1,3,5-triazin-2-one

Summary for 4Q4M
Entry DOI10.2210/pdb4q4m/pdb
Related4Q4O 4Q4P 4Q4Q 4Q4R 4Q4S
DescriptorQueuine tRNA-ribosyltransferase, ZINC ION, 6-amino-4-phenyl-1,3,5-triazin-2(1H)-one, ... (5 entities in total)
Functional Keywordstransferase, preq1, trna, guanine exchange enzyme, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceZymomonas mobilis subsp. mobilis
Total number of polymer chains1
Total formula weight43491.83
Authors
Neeb, M.,Heine, A.,Klebe, G. (deposition date: 2014-04-15, release date: 2015-06-10, Last modification date: 2023-09-20)
Primary citationNeeb, M.,Hohn, C.,Heine, A.,Diederich, F.,Klebe, G.
5-Azacytosines as a Novel Scaffold to Inhibit Z. mobilis TGT with Expected Improved Bioavailability and Synthetic Accessibility
To be Published,
Experimental method
X-RAY DIFFRACTION (1.621 Å)
Structure validation

217705

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