4KRS
Tankyrase-1 complexed with small molecule inhibitor
Summary for 4KRS
Entry DOI | 10.2210/pdb4krs/pdb |
Descriptor | Tankyrase-1, ZINC ION, SULFATE ION, ... (5 entities in total) |
Functional Keywords | transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm: O95271 |
Total number of polymer chains | 2 |
Total formula weight | 51921.24 |
Authors | |
Primary citation | Shultz, M.D.,Majumdar, D.,Chin, D.N.,Fortin, P.D.,Feng, Y.,Gould, T.,Kirby, C.A.,Stams, T.,Waters, N.J.,Shao, W. Structure-Efficiency Relationship of [1,2,4]Triazol-3-ylamines as Novel Nicotinamide Isosteres that Inhibit Tankyrases. J.Med.Chem., 56:7049-7059, 2013 Cited by PubMed: 23879431DOI: 10.1021/jm400826j PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.29 Å) |
Structure validation
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