Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

4KRS

Tankyrase-1 complexed with small molecule inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 1401
ChainResidue
ACYS1234
AHIS1237
ACYS1242
ACYS1245

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1402
ChainResidue
AHIS1132
AARG1133
ALYS1220
AALA1288
AHOH1540

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1403
ChainResidue
AHIS1176
AHOH1534
BHIS1176
BHIS1177
BASN1178

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1404
ChainResidue
AASN1143
AARG1144
APRO1313
AGLU1314
AHOH1504

site_idAC5
Number of Residues2
DetailsBINDING SITE FOR RESIDUE SO4 A 1405
ChainResidue
AARG1149
AHIS1246

site_idAC6
Number of Residues9
DetailsBINDING SITE FOR RESIDUE 1SX A 1406
ChainResidue
AHIS1184
AGLY1185
ASER1186
APHE1188
ATYR1203
ATYR1213
ASER1221
ATYR1224
AHOH1537

site_idAC7
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN B 1401
ChainResidue
BCYS1234
BHIS1237
BCYS1242
BCYS1245

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 B 1402
ChainResidue
BARG1130
BHIS1132
BARG1133
BLYS1220
BHOH1502

site_idAC9
Number of Residues9
DetailsBINDING SITE FOR RESIDUE 1SX B 1403
ChainResidue
BHIS1184
BGLY1185
BPHE1188
BTYR1203
BTYR1213
BSER1221
BTYR1224
BILE1228
BHOH1551

221051

PDB entries from 2024-06-12

PDB statisticsPDBj update infoContact PDBjnumon