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4GL9

Crystal structure of inhibitory protein SOCS3 in complex with JAK2 kinase domain and fragment of GP130 intracellular domain

4GL9 の概要
エントリーDOI10.2210/pdb4gl9/pdb
分子名称Tyrosine-protein kinase, Interleukin-6 receptor subunit beta, Suppressor of cytokine signaling 3,Suppressor of cytokine signaling 3,Suppressor of cytokine signaling 3,Suppressor of cytokine signaling 3, ... (5 entities in total)
機能のキーワードkinase inhibitor receptor cytokine signalling, phosphorylation, transferase-transferase inhibitor complex, transferase/transferase inhibitor
由来する生物種Mus musculus (Mouse)
詳細
タンパク質・核酸の鎖数12
化学式量合計210768.17
構造登録者
Kershaw, N.J.,Murphy, J.M.,Laktyushin, A.,Nicola, N.A.,Babon, J.J. (登録日: 2012-08-14, 公開日: 2013-03-06, 最終更新日: 2018-06-13)
主引用文献Kershaw, N.J.,Murphy, J.M.,Liau, N.P.,Varghese, L.N.,Laktyushin, A.,Whitlock, E.L.,Lucet, I.S.,Nicola, N.A.,Babon, J.J.
SOCS3 binds specific receptor-JAK complexes to control cytokine signaling by direct kinase inhibition.
Nat.Struct.Mol.Biol., 20:469-476, 2013
Cited by
PubMed: 23454976
DOI: 10.1038/nsmb.2519
主引用文献が同じPDBエントリー
実験手法
X-RAY DIFFRACTION (3.9 Å)
構造検証レポート
Validation report summary of 4gl9
検証レポート(詳細版)ダウンロードをダウンロード

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件を2024-03-27に公開中

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