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4C68

Plasmodium vivax N-myristoyltransferase in complex with a peptidomimetic inhibitor

Summary for 4C68
Entry DOI10.2210/pdb4c68/pdb
Related4C7H 4C7I
DescriptorGLYCYLPEPTIDE N-TETRADECANOYLTRANSFERASE, FORMIC ACID, DIMETHYL SULFOXIDE, ... (9 entities in total)
Functional Keywordstransferase, myristoylation, malaria
Biological sourcePLASMODIUM VIVAX
Total number of polymer chains3
Total formula weight139621.37
Authors
Olaleye, T.O.,Brannigan, J.A.,Goncalves, V.,Roberts, S.M.,Leatherbarrow, R.J.,Wilkinson, A.J.,Tate, E.W. (deposition date: 2013-09-17, release date: 2014-09-24, Last modification date: 2024-05-08)
Primary citationOlaleye, T.O.,Brannigan, J.A.,Roberts, S.M.,Leatherbarrow, R.J.,Wilkinson, A.J.,Tate, E.W.
Peptidomimetic Inhibitors of N-Myristoyltransferase from Human Malaria and Leishmaniasis Parasites.
Org.Biomol.Chem., 12:8132-, 2014
Cited by
PubMed: 25230674
DOI: 10.1039/C4OB01669F
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.38 Å)
Structure validation

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