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4BZB

Crystal structure of the tetrameric dGTP-bound SAMHD1 mutant catalytic core

Summary for 4BZB
Entry DOI10.2210/pdb4bzb/pdb
Related4BZC
DescriptorDEOXYNUCLEOSIDE TRIPHOSPHATE TRIPHOSPHOHYDROLASE SAMHD1, 2'-DEOXYGUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ... (4 entities in total)
Functional Keywordshydrolase, hiv restriction factor, dntpase
Biological sourceHOMO SAPIENS (HUMAN)
Total number of polymer chains4
Total formula weight259986.11
Authors
Ji, X.,Yang, H.,Wu, Y.,Yan, J.,Mehrens, J.,DeLucia, M.,Hao, C.,Gronenborn, A.M.,Skowronski, J.,Ahn, J.,Xiong, Y. (deposition date: 2013-07-25, release date: 2013-10-23, Last modification date: 2023-12-20)
Primary citationJi, X.,Wu, Y.,Yan, J.,Mehrens, J.,Yang, H.,Delucia, M.,Hao, C.,Gronenborn, A.M.,Skowronski, J.,Ahn, J.,Xiong, Y.
Mechanism of Allosteric Activation of Samhd1 by Dgtp
Nat.Struct.Mol.Biol., 20:1304-, 2013
Cited by
PubMed: 24141705
DOI: 10.1038/NSMB.2692
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.83 Å)
Structure validation

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