4PNI
Bovine G protein-coupled receptor kinase 1 in complex with GSK2163632A
Summary for 4PNI
Entry DOI | 10.2210/pdb4pni/pdb |
Related | 4L9I 4PNK |
Descriptor | Rhodopsin kinase, 3-[(2-{[1-(N,N-dimethylglycyl)-6-methoxy-4,4-dimethyl-1,2,3,4-tetrahydroquinolin-7-yl]amino}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]thiophene-2-carboxamide, CHLORIDE ION, ... (4 entities in total) |
Functional Keywords | agc family kinase, ser/thr kinase, rgs homology domain, g protein coupled receptor kinase, grk, grk1, rhodopsin kinase, hydrolyase, gpcr, phosphorylation, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Bos taurus (Bovine) |
Total number of polymer chains | 1 |
Total formula weight | 63773.20 |
Authors | Homan, K.T.,Tesmer, J.J.G. (deposition date: 2014-05-23, release date: 2014-10-08, Last modification date: 2023-12-27) |
Primary citation | Homan, K.T.,Larimore, K.M.,Elkins, J.M.,Szklarz, M.,Knapp, S.,Tesmer, J.J. Identification and structure-function analysis of subfamily selective g protein-coupled receptor kinase inhibitors. Acs Chem.Biol., 10:310-319, 2015 Cited by PubMed: 25238254DOI: 10.1021/cb5006323 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.85 Å) |
Structure validation
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