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4NP3

Crystal structure of the murine cd44 hyaluronan binding domain complex with a small molecule

Summary for 4NP3
Entry DOI10.2210/pdb4np3/pdb
Related4MRD 4MRE 4MRF 4MRG 4MRH 4NP2
DescriptorCD44 antigen, 2-[(4-methyl-1H-imidazol-5-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-8-amine, DIMETHYL SULFOXIDE, ... (6 entities in total)
Functional Keywordslink module, cell surface receptor, hyaluronan, non-glycosylated, cell surface, cell adhesion-inhibitor complex, cell adhesion/inhibitor
Biological sourceMus musculus (mouse)
Cellular locationCell membrane; Single-pass type I membrane protein: P15379
Total number of polymer chains1
Total formula weight17528.48
Authors
Liu, L.K.,Finzel, B. (deposition date: 2013-11-20, release date: 2014-04-16)
Primary citationLiu, L.K.,Finzel, B.C.
Fragment-Based Identification of an Inducible Binding Site on Cell Surface Receptor CD44 for the Design of Protein-Carbohydrate Interaction Inhibitors.
J.Med.Chem., 57:2714-2725, 2014
Cited by
PubMed: 24606063
DOI: 10.1021/jm5000276
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.61 Å)
Structure validation

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