3PUH
Cocaine Esterase, wild-type biologically active dimer
Summary for 3PUH
Entry DOI | 10.2210/pdb3puh/pdb |
Related | 1ju3 1ju4 3i2f 3i2g 3i2h 3i2i 3i2j 3ida 3PUI |
Descriptor | Cocaine esterase, GLYCEROL, SULFATE ION, ... (4 entities in total) |
Functional Keywords | alpha/beta hydrolase, jelly-roll beta-barrel, cleavage of cocaine, hydrolase |
Biological source | Rhodococcus sp. |
Cellular location | Cytoplasm : Q9L9D7 |
Total number of polymer chains | 2 |
Total formula weight | 128080.72 |
Authors | Nance, M.R.,Tesmer, J.J.G. (deposition date: 2010-12-04, release date: 2011-09-21, Last modification date: 2024-02-21) |
Primary citation | Narasimhan, D.,Collins, G.T.,Nance, M.R.,Nichols, J.,Edwald, E.,Chan, J.,Ko, M.C.,Woods, J.H.,Tesmer, J.J.,Sunahara, R.K. Subunit stabilization and polyethylene glycolation of cocaine esterase improves in vivo residence time. Mol.Pharmacol., 80:1056-1065, 2011 Cited by PubMed: 21890748DOI: 10.1124/mol.111.074997 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.3 Å) |
Structure validation
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