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3MY1

Structure of CDK9/cyclinT1 in complex with DRB

Summary for 3MY1
Entry DOI10.2210/pdb3my1/pdb
Related3BLH 3BLQ 3BLR 3MY5
DescriptorCell division protein kinase 9, Cyclin-T1, PHOSPHATE ION, ... (6 entities in total)
Functional Keywordscdk-cyclin complex, phosphorylated, transcription-protein binding-inhibitor complex, transcription/protein binding/inhibitor
Biological sourceHomo sapiens (human)
More
Cellular locationNucleus: P50750 O60563
Total number of polymer chains2
Total formula weight69048.09
Authors
Baumli, S.,Johnson, L.N. (deposition date: 2010-05-09, release date: 2010-09-29, Last modification date: 2023-11-01)
Primary citationBaumli, S.,Endicott, J.A.,Johnson, L.N.
Halogen bonds form the basis for selective P-TEFb inhibition by DRB
Chem.Biol., 17:931-936, 2010
Cited by
PubMed: 20851342
DOI: 10.1016/j.chembiol.2010.07.012
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.8 Å)
Structure validation

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