3E94
Crystal structure of RXRalpha ligand binding domain in complex with tributyltin and a coactivator fragment
Summary for 3E94
Entry DOI | 10.2210/pdb3e94/pdb |
Related | 1LBD 1XDK 2P1T 2P1U 2P1V |
Descriptor | Retinoic acid receptor RXR-alpha, Nuclear receptor coactivator 2 peptide, tributylstannanyl, ... (5 entities in total) |
Functional Keywords | protein-ligand complex, dna-binding, host-virus interaction, metal-binding, nucleus, polymorphism, receptor, transcription, transcription regulation, ubl conjugation, zinc, zinc-finger, activator, phosphoprotein |
Biological source | Homo sapiens (human) More |
Cellular location | Nucleus: P19793 Q15596 |
Total number of polymer chains | 2 |
Total formula weight | 29198.48 |
Authors | Bourguet, W.,Le Maire, A. (deposition date: 2008-08-21, release date: 2009-03-10, Last modification date: 2023-08-30) |
Primary citation | le Maire, A.,Grimaldi, M.,Roecklin, D.,Dagnino, S.,Vivat-Hannah, V.,Balaguer, P.,Bourguet, W. Activation of RXR-PPAR heterodimers by organotin environmental endocrine disruptors Embo Rep., 10:367-373, 2009 Cited by PubMed: 19270714DOI: 10.1038/embor.2009.8 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.9 Å) |
Structure validation
Download full validation report