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3BHH

Crystal structure of human calcium/calmodulin-dependent protein kinase IIB isoform 1 (CAMK2B)

Summary for 3BHH
Entry DOI10.2210/pdb3bhh/pdb
DescriptorCalcium/calmodulin-dependent protein kinase type II beta chain, [4-({4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrile (3 entities in total)
Functional Keywordscamk2b, cam2, camk2, cam kinase ii beta chain, camk ii beta subunit, calcium/calmodulion dependent protein kinase ii beta, ec:2.7.1.123, mgc29528, proline rich calmodulin dependent protein kinase, structural genomics consortium, sgc, atp-binding, calmodulin-binding, nucleotide-binding, phosphoprotein, serine/threonine-protein kinase, transferase
Biological sourceHomo sapiens (human)
Total number of polymer chains4
Total formula weight134979.33
Authors
Primary citationFilippakopoulos, P.,Rellos, P.,Niesen, F.,Burgess, N.,Bullock, A.,Berridge, G.,Pike, A.C.W.,Ugochukwu, E.,Pilka, E.S.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Weigelt, J.,Knapp, S.
Crystal Structure of Human Calcium/Calmodulin-Dependent Protein Kinase IIB Isoform 1 (CAMK2B).
To be Published,
Experimental method
X-RAY DIFFRACTION (2.4 Å)
Structure validation

217705

PDB entries from 2024-03-27

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