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3AQV

Human AMP-activated protein kinase alpha 2 subunit kinase domain (T172D) complexed with compound C

3AQV の概要
エントリーDOI10.2210/pdb3aqv/pdb
関連するPDBエントリー2h6d 2yza
分子名称5'-AMP-activated protein kinase catalytic subunit alpha-2, 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine (3 entities in total)
機能のキーワードstructural genomics, riken structural genomics/proteomics initiative, rsgi, transferase, signaling protein, serine/threonine protein kinase, phosphorylation, atp-binding, nucleotide-binding, cholesterol biosynthesis, fatty acid biosynthesis, lipid synthesis, glucose metabolism, magnesium, metal-binding, serine/threonine-protein kinase, steroid biosynthesis, transferase-transferase inhibitor complex, transferase/transferase inhibitor
由来する生物種Homo sapiens (human)
細胞内の位置Cytoplasm (By similarity): P54646
タンパク質・核酸の鎖数1
化学式量合計31971.22
構造登録者
主引用文献Handa, N.,Takagi, T.,Saijo, S.,Kishishita, S.,Takaya, D.,Toyama, M.,Terada, T.,Shirouzu, M.,Suzuki, A.,Lee, S.,Yamauchi, T.,Okada-Iwabu, M.,Iwabu, M.,Kadowaki, T.,Minokoshi, Y.,Yokoyama, S.
Structural basis for compound C inhibition of the human AMP-activated protein kinase alpha 2 subunit kinase domain
Acta Crystallogr.,Sect.D, 67:480-487, 2011
Cited by
PubMed: 21543851
DOI: 10.1107/S0907444911010201
主引用文献が同じPDBエントリー
実験手法
X-RAY DIFFRACTION (2.08 Å)
構造検証レポート
Validation report summary of 3aqv
検証レポート(詳細版)ダウンロードをダウンロード

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件を2024-09-18に公開中

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