3MVJ
Human cyclic AMP-dependent protein kinase PKA inhibitor complex
Summary for 3MVJ
Entry DOI | 10.2210/pdb3mvj/pdb |
Related | 3MV5 3MVH |
Descriptor | cAMP-dependent protein kinase catalytic subunit alpha, cAMP-dependent protein kinase inhibitor alpha, (3R)-1-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine, ... (4 entities in total) |
Functional Keywords | kinase inhibitor, transferase |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm. Isoform 2: Cell projection, cilium, flagellum : P17612 |
Total number of polymer chains | 6 |
Total formula weight | 136053.52 |
Authors | Pandit, J.,Vajdos, F. (deposition date: 2010-05-04, release date: 2010-06-02, Last modification date: 2017-11-08) |
Primary citation | Freeman-Cook, K.D.,Autry, C.,Borzillo, G.,Gordon, D.,Barbacci-Tobin, E.,Bernardo, V.,Briere, D.,Clark, T.,Corbett, M.,Jakubczak, J.,Kakar, S.,Knauth, E.,Lippa, B.,Luzzio, M.J.,Mansour, M.,Martinelli, G.,Marx, M.,Nelson, K.,Pandit, J.,Rajamohan, F.,Robinson, S.,Subramanyam, C.,Wei, L.,Wythes, M.,Morris, J. Design of selective, ATP-competitive inhibitors of Akt. J.Med.Chem., 53:4615-4622, 2010 Cited by PubMed: 20481595DOI: 10.1021/jm1003842 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.49 Å) |
Structure validation
Download full validation report