3BHV
Structure of phosphorylated Thr160 CDK2/cyclin A in complex with the inhibitor variolin B
Summary for 3BHV
Entry DOI | 10.2210/pdb3bhv/pdb |
Related | 3BHT 3BHU |
Descriptor | Cell division protein kinase 2, Cyclin-A2, 9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-ol, ... (6 entities in total) |
Functional Keywords | ser/thr protein kinase, transferase, phosphorylation, cell cycle, atp-binding, cell division, mitosis, nucleotide-binding, phosphoprotein, polymorphism, serine/threonine-protein kinase, cyclin |
Biological source | Homo sapiens (human) More |
Cellular location | Nucleus: P30274 |
Total number of polymer chains | 4 |
Total formula weight | 129398.12 |
Authors | Echalier, A.,Bettayeb, K.,Ferandin, Y.,Lozach, O.,Clement, M.,Valette, A.,Liger, F.,Marquet, B.,Morris, J.C.,Endicott, J.A.,Joseph, B.,Meijer, L. (deposition date: 2007-11-29, release date: 2008-02-12, Last modification date: 2011-07-13) |
Primary citation | Bettayeb, K.,Tirado, O.M.,Marionneau-Lambot, S.,Ferandin, Y.,Lozach, O.,Morris, J.C.,Mateo-Lozano, S.,Drueckes, P.,Kubbutat, M.H.,Liger, F.,Marquet, B.,Joseph, B.,Echalier, A.,Endicott, J.A.,Notario, V.,Meijer, L. Meriolins, a new class of cell death inducing kinase inhibitors with enhanced selectivity for cyclin-dependent kinases Cancer Res., 67:8325-8334, 2007 Cited by PubMed: 17804748DOI: 10.1158/0008-5472.CAN-07-1826 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
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