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2XUF

CRYSTAL STRUCTURE OF MACHE-Y337A-TZ2PA6 ANTI COMPLEX (1 MTH)

Summary for 2XUF
Entry DOI10.2210/pdb2xuf/pdb
Related1C2B 1C2O 1J06 1J07 1KU6 1MAA 1MAH 1N5M 1N5R 1Q83 1Q84 2C0P 2C0Q 2H9Y 2HA0 2HA2 2HA3 2HA4 2HA5 2HA6 2HA7 2JEY 2JEZ 2JF0 2JGE 2JGF 2JGG 2JGH 2JGI 2JGJ 2JGK 2JGL 2JGM 2WHP 2WHQ 2WHR 2WLS 2WU3 2WU4 2XUD 2XUG 2XUH 2XUI 2XUJ 2XUK 2XUO 2XUP
DescriptorACETYLCHOLINESTERASE, 2-acetamido-2-deoxy-beta-D-glucopyranose, HEXAETHYLENE GLYCOL, ... (5 entities in total)
Functional Keywordshydrolase, hydrolase fold, femtomolar inhibitor, click chemistry
Biological sourceMUS MUSCULUS (HOUSE MOUSE)
Total number of polymer chains2
Total formula weight121535.41
Authors
Bourne, Y.,Radic, Z.,Taylor, P.,Marchot, P. (deposition date: 2010-10-19, release date: 2010-12-08, Last modification date: 2023-12-20)
Primary citationBourne, Y.,Radic, Z.,Taylor, P.,Marchot, P.
Conformational Remodeling of Femtomolar Inhibitor-Acetylcholinesterase Complexes in the Crystalline State
J.Am.Chem.Soc., 132:18292-, 2010
Cited by
PubMed: 21090615
DOI: 10.1021/JA106820E
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.55 Å)
Structure validation

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