2DTZ
Crystal Structure of multidrug binding protein QacR from Staphylococcus aureus cocrystallized with compound DB75
Summary for 2DTZ
Entry DOI | 10.2210/pdb2dtz/pdb |
Related | 1JT6 1RKW 1RPW 2HQ5 |
Descriptor | HTH-type transcriptional regulator qacR, SULFATE ION (3 entities in total) |
Functional Keywords | multidrug recognition, db75, qacr, multidrug binding protein, transcription |
Biological source | Staphylococcus aureus |
Total number of polymer chains | 4 |
Total formula weight | 92700.60 |
Authors | Brooks, B.E.,Brennan, R.G. (deposition date: 2006-07-19, release date: 2007-07-17, Last modification date: 2023-10-25) |
Primary citation | Brooks, B.E.,Piro, K.M.,Brennan, R.G. Multidrug-Binding Transcription Factor QacR Binds the Bivalent Aromatic Diamidines DB75 and DB359 in Multiple Positions J.Am.Chem.Soc., 129:8389-8395, 2007 Cited by PubMed: 17567017DOI: 10.1021/ja072576v PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
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