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1T65

Crystal structure of the androgen receptor ligand binding domain with DHT and a peptide derived form its physiological coactivator GRIP1 NR box 2 bound in a non-helical conformation

Summary for 1T65
Entry DOI10.2210/pdb1t65/pdb
Related1T5Z 1T63
DescriptorAndrogen receptor, Nuclear receptor coactivator 2, 5-ALPHA-DIHYDROTESTOSTERONE, ... (4 entities in total)
Functional Keywordsandrogen receptor ligand binding domain grip1 nr box2 coactivators crystal structure non-helical, hormone-growth factor complex, hormone/growth factor
Biological sourceHomo sapiens (human)
More
Cellular locationNucleus : P10275 Q15596
Total number of polymer chains2
Total formula weight31147.65
Authors
Estebanez-Perpina, E.,Moore, J.M.R.,Mar, E.,Nguyen, P.,Delgado-Rodrigues, E.,Baxter, J.D.,Webb, P.,Fletterick, R.J.,Guy, R.K. (deposition date: 2004-05-05, release date: 2005-01-25, Last modification date: 2024-02-14)
Primary citationEstebanez-Perpina, E.,Moore, J.M.R.,Mar, E.,Delgado-Rodrigues, E.,Nguyen, P.,Baxter, J.D.,Buehrer, B.M.,Webb, P.,Fletterick, R.J.,Guy, R.K.
The Molecular Mechanisms of Coactivator Utilization in Ligand-dependent Transactivation by the Androgen Receptor.
J.Biol.Chem., 280:8060-8068, 2005
Cited by
PubMed: 15563469
DOI: 10.1074/jbc.M407046200
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.66 Å)
Structure validation

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