1OVE
The structure of p38 alpha in complex with a dihydroquinolinone
Summary for 1OVE
Entry DOI | 10.2210/pdb1ove/pdb |
Related | 1M7Q 1OUK 1OUY |
Descriptor | Mitogen-activated protein kinase 14, 1-(2,6-DICHLOROPHENYL)-5-(2,4-DIFLUOROPHENYL)-7-PIPERIDIN-4-YL-3,4-DIHYDROQUINOLIN-2(1H)-ONE, GLYCEROL, ... (4 entities in total) |
Functional Keywords | map kinase, hydrophobic pocket, kinase domain, linker region, transferase |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm (By similarity): Q16539 |
Total number of polymer chains | 1 |
Total formula weight | 42562.33 |
Authors | Fitzgerald, C.E.,Patel, S.B.,Becker, J.W.,Cameron, P.M.,Zaller, D.,Pikounis, V.B.,O'Keefe, S.J.,Scapin, G. (deposition date: 2003-03-26, release date: 2003-09-02, Last modification date: 2023-08-16) |
Primary citation | Fitzgerald, C.E.,Patel, S.B.,Becker, J.W.,Cameron, P.M.,Zaller, D.,Pikounis, V.B.,O'Keefe, S.J.,Scapin, G. Structural basis for p38alpha MAP kinase quinazolinone and pyridol-pyrimidine inhibitor specificity Nat.Struct.Biol., 10:764-769, 2003 Cited by PubMed: 12897767DOI: 10.1038/nsb949 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
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